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HuagongsheHuagongshe Chemie-Druckbericht · Nur für Forschungszwecke
HRID 1979330Erstellt: 24. Oktober 2026

Cyclopentanecarbonyl chloride → 2-oxo-3-tert-butoxycarbonylamino-5-cyclopentylcarbonyl-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepine

https://huagongshe.com/de/reaction/1979330

Reaktionsgleichung

Beteiligte Stoffe

RolleNameHCIDEinwaage
EduktCyclopentanecarbonyl chlorideHCID 78284—
EduktHCID 15490831HCID 15490831—
Edukt2-oxo-3-tert-butoxycarbonylamino-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepineHCID 21201581—
Produkt2-oxo-3-tert-butoxycarbonylamino-5-cyclopentylcarbonyl-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepineHCID 21201645—

Reaktionsschritte

Step 1 of Example 1 was repeated except that cyclopentylcarbonyl chloride was used instead of pivaloyl chloride, and that 2-oxo-3-tert-butoxycarbonylamino-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepine obtained from Referential Example 4 was used instead of 2-oxo-3-tert-butoxycarbonylamino-1,3,4,5-tetrahydro-2H-1,5-benzodiazepine, to thereby obtain the title compound.

Herkunft & Nachweise

DOI10.6084/m9.figshare.5104873.v1
PatentnummerUS06239131B1
Quelldatensatzuspto-grants-2001_05
ORD IDord-2e9220b093cb4c93864b1382bb275986
Quellennotizuspto-grants-2001_05