5-(5,6-difluoro1H-indol-2-yl)-2-methoxy-phenylamine → (4-{3-[5-(5,6-Difluoro-1h-indol-2-yl)-2-methoxy-phenyl]-thioureido}-benzyl)-phosphonic acid diethyl ester

Beteiligte Stoffe

Reaktionsschritte

The product from Example 3, 5-(5,6-difluoro-1H-indol-2-yl)-2-methoxy-phenylamine, (0.137 g, 0.5 mmol) was reacted with the product from Example 23, Step A (0.156 g, 0.54 mmol) according to the procedure for Example 23, Step B to give the product (0.172 g), mp 180-182° C.

Herkunft & Nachweise