2-Oxoimidazolidine-1-carbonyl chloride → cis-4-(3-Chloro-4-methoxy-phenyl)-2-{1-[1-(2-oxo-imidazolidin-1-yl)-methanoyl]-piperidin-4-yl}-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one

関与物質

役割	名称	HCID	仕込み量
反応物	2-Oxoimidazolidine-1-carbonyl chloride	HCID 83241	—
反応物	(cis)-4-(3-Chloro-4-methoxy-phenyl)-2-[1-(1-morpholin-4-yl-methanoyl)-piperidin-4-yl]-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one	HCID 69490073	—
生成物	cis-4-(3-Chloro-4-methoxy-phenyl)-2-{1-[1-(2-oxo-imidazolidin-1-yl)-methanoyl]-piperidin-4-yl}-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one	HCID 69487067	—

Prepared from intermediate product A1 and 2-oxo-imidazolidine-1-carbonyl chloride as described for compound 1. M. p. 216–218° C.