2-(Chloromethyl)-2,3-dihydro-1,4-benzodioxin → {5-Chloro-3-[3-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-4-oxo-3,4-dihydro-phthalazin-1-yl]-2-methyl-indol-1-yl}-acetic acid

Beteiligte Stoffe

Rolle	Name	HCID	Einwaage
Edukt	2-(Chloromethyl)-2,3-dihydro-1,4-benzodioxin	HCID 95320	—
Edukt	tert-butyl 2-(5-chloro-3-(4-hydroxyphthalazin-1-yl)-2-methyl-1H-indol-1-yl)acetate	HCID 58247168	—
Produkt	{5-Chloro-3-[3-(2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-4-oxo-3,4-dihydro-phthalazin-1-yl]-2-methyl-indol-1-yl}-acetic acid	HCID 11706240	—

Reaktionsschritte

The title compound was prepared from the product of example 16, step c) and 2-chloromethyl-2,3-dihydro-benzo[1,4]dioxine using the procedure described in example 14. MS: ESI (negative): 514, 516 (M−H).

Herkunft & Nachweise

DOI	10.6084/m9.figshare.5104873.v1
Patentnummer	US07981912B2
Quelldatensatz	uspto-grants-2011_07
ORD ID	ord-c0bce16399494bdab37d68e948f49aa3
Quellennotiz	uspto-grants-2011_07