1-Cyclopropyl-1-(5-methyl-1,2,4-oxadiazol-3-yl)ethan-1-amine → 5-Cyclopropyl-4-cyclopropylmethoxy-pyridine-2-carboxylic acid [1-cyclopropyl-1-(5-methyl-[1,2,4]oxadiazol-3-yl)-ethyl]-amide

Beteiligte Stoffe

Rolle	Name	HCID	Einwaage
Edukt	1-Cyclopropyl-1-(5-methyl-1,2,4-oxadiazol-3-yl)ethan-1-amine	HCID 43559223	—
Edukt	5-Cyclopropyl-4-cyclopropylmethoxy-pyridine-2-carboxylic acid	HCID 90203809	—
Produkt	5-Cyclopropyl-4-cyclopropylmethoxy-pyridine-2-carboxylic acid [1-cyclopropyl-1-(5-methyl-[1,2,4]oxadiazol-3-yl)-ethyl]-amide	HCID 76282968	—

Reaktionsschritte

The title compound was synthesized in analogy to Example 24d, using 5-Cyclopropyl-4-cyclopropylmethoxy-pyridine-2-carboxylic acid (Example 42c) and 1-Cyclopropyl-1-(5-methyl-[1,2,4]oxadiazol-3-yl)-ethylamine (CAN 1155536-64-3) as starting materials and isolated (13 mg, 23%) as colorless oil; MS (ESI, m/z): 383.6 (M+H+)

Herkunft & Nachweise

DOI	10.6084/m9.figshare.5104873.v1
Patentnummer	US09409866B2
Quelldatensatz	uspto-grants-2016_08
ORD ID	ord-c213e5fa60d44cf0b6306ced0f696d87
Quellennotiz	uspto-grants-2016_08