Zurück
HuagongsheHuagongshe Chemie-Druckbericht · Nur für Forschungszwecke
HRID 1665791Erstellt: 26. Oktober 2026

5,8,14-Triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2,4,6,8,10-pentaene → p-Toluenesulfonic acid

https://huagongshe.com/reaction/1665791

Reaktionsgleichung

Beteiligte Stoffe

RolleNameHCIDEinwaage
Edukt5,8,14-Triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2,4,6,8,10-pentaeneHCID 170361—
EduktVarenicline TosylateHCID 86637773—
Produktp-Toluenesulfonic acidHCID 6101—

Reaktionsschritte

Varenicline Tosylate can be prepared by combining Varenicline base, a solvent and p-Toluene sulfonic acid (p-TSA) to obtain a reaction mixture and precipitating Varenicline Tosylate from the reaction mixture. Preferably, the obtained Varenicline Tosylate is further recovered from the reaction mixture.

Herkunft & Nachweise

DOI10.6084/m9.figshare.5104873.v1
PatentnummerUS08039620B2
Quelldatensatzuspto-grants-2011_10
ORD IDord-a043c6acb8064c67afa11162b50f2adf
Quellennotizuspto-grants-2011_10