(4-(Methylsulfinyl)phenyl)boronic acid → (3-Fluoro-4'-methanesulfinyl-biphenyl-4-yl)-(2-(S)-pyrrolidin-1-ylmethyl-pyrrolidin-1-yl)-methanone

Beteiligte Stoffe

Rolle	Name	HCID	Einwaage
Edukt	(4-(Methylsulfinyl)phenyl)boronic acid	HCID 2773531	—
Edukt	(4-Bromo-2-fluoro-phenyl)-((S)-2-pyrrolidin-1-ylmethyl-pyrrolidin-1-yl)-methanone	HCID 11965125	—
Produkt	(3-Fluoro-4'-methanesulfinyl-biphenyl-4-yl)-(2-(S)-pyrrolidin-1-ylmethyl-pyrrolidin-1-yl)-methanone	HCID 57980145	—

Reaktionsschritte

The title compound is prepared in a manner substantially analogous to Procedure SS starting from (4-bromo-2-fluoro-phenyl)-(2-(S)-pyrrolidin-1-ylmethyl-pyrrolidin-1-yl)-methanone and 4-Methylsulfinyl benzene boronic acid. MS (M+H) 415.1

Herkunft & Nachweise

DOI	10.6084/m9.figshare.5104873.v1
Patentnummer	US07632857B2
Quelldatensatz	uspto-grants-2009_12
ORD ID	ord-3ca7ad54580b4f07bb19f0070e6e7030
Quellennotiz	uspto-grants-2009_12