3-Bromopyridine → 6-pyridin-3-yl-1H-indole
Reaktionsgleichung
COC1C=CC(B(O)O)=CC=1.Br[C:13]1[CH:14]=[N:15][CH:16]=[CH:17][CH:18]=1.C(OC([N:26]1[C:34]2[C:29](=[CH:30][CH:31]=[C:32](Br)[CH:33]=2)[CH:28]=[CH:27]1)=O)(C)(C)C>>[N:15]1[CH:16]=[CH:17][CH:18]=[C:13]([C:32]2[CH:33]=[C:34]3[C:29]([CH:28]=[CH:27][NH:26]3)=[CH:30][CH:31]=2)[CH:14]=1Komponenten
4
Versuchsvorschrift
The desired compound was prepared according to the method of Example 25, step 1, except substituting 6-indolylboronic acid, prepared as in step 1 for 4-methoxyphenylboronic acid, and 3-bromopyridine for 1-tert-butoxycarbonyl-6-bromoindole.
Quellen und Nachweise
- ORD-Eintrag
- ord-721e837f50e24c1185023a93de50dbe0
- Quelldatensatz
- uspto-grants-1995_10
- Patentnummer
- US05459152
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