5-Isocyanato-1,2,3-trimethoxybenzene → 1-[2-(phenyl)-2-(3,4,5-trimethoxyphenylcarbamoyloxy)ethyl]4-(6-fluoro-1-methyl-1H-indazol-3-yl)piperidine

Beteiligte Stoffe

Reaktionsschritte

Starting from 1-(2-hydroxy-2-phenyl-ethyl)-4-(6-fluoro-1-methyl-1H -indazol-3-yl)-piperidine (300 mg; 0.85 mmol) and 3,4,5-trimethoxyphenylisocyanate (300 mg; 1.44 mmol) using the procedure described in example 8B was prepared 160 mg (34%) of the title compound.

Herkunft & Nachweise