(2-Methyl-1,3-thiazol-4-yl)acetic acid → HCID 58349704, Verbindung
Reaktionsgleichung
[CH3:1][C:2]1[S:3][CH:4]=[C:5]([CH2:7][C:8]([OH:10])=O)[N:6]=1.[CH3:11][NH:12][C@H:13]1[CH2:32][N:17]2[C:18]3[C:23]([C:24]([CH2:25][C:26]([O:28]CCC)=[O:27])=[C:16]2[CH2:15][CH2:14]1)=[CH:22][CH:21]=[CH:20][CH:19]=3>>[CH3:11][N:12]([C:8](=[O:10])[CH2:7][C:5]1[N:6]=[C:2]([CH3:1])[S:3][CH:4]=1)[C@H:13]1[CH2:32][N:17]2[C:18]3[C:23]([C:24]([CH2:25][C:26]([OH:28])=[O:27])=[C:16]2[CH2:15][CH2:14]1)=[CH:22][CH:21]=[CH:20][CH:19]=3Komponenten
3
Versuchsvorschrift
The title compound was prepared using analogous procedures described in Example 1 (Method A) from (2-methyl-1,3-thiazol-4-yl)acetic acid and propyl [(7R)-7-(methylamino)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl]acetate. MS (+ESI) m/z: 398.
Quellen und Nachweise
- ORD-Eintrag
- ord-cd91c22ed154410b9745b92d1771f378
- Quelldatensatz
- uspto-grants-2014_01