Methyl 4-aminobenzoate → Methyl 4-({2-[4-(2-bromo-5-chlorophenyl)-2-oxopyridin-1(2H)-yl]-3-(pyridin-3-yl)propanoyl}amino)benzoate

Beteiligte Stoffe

Rolle	Name	HCID	Einwaage
Edukt	Methyl 4-aminobenzoate	HCID 12082	—
Edukt	2-[4-(2-Bromo-5-chlorophenyl)-2-oxopyridin-1(2H)-yl]-3-(pyridin-3-yl)propanoic acid	HCID 117622698	—
Produkt	Methyl 4-({2-[4-(2-bromo-5-chlorophenyl)-2-oxopyridin-1(2H)-yl]-3-(pyridin-3-yl)propanoyl}amino)benzoate	HCID 117622651	—

Reaktionsschritte

244 mg (purity 57%, 0.32 mmol) of 2-[4-(2-bromo-5-chlorophenyl)-2-oxopyridin-1(2H)-yl]-3-(pyridin-3-yl)propanoic acid (racemate) and 1.2 eq. of methyl 4-aminobenzoate were reacted according to General Method 5A. Yield: 65 mg (purity 85%, 30% of theory)

Herkunft & Nachweise

DOI	10.6084/m9.figshare.5104873.v1
Patentnummer	US09434690B2
Quelldatensatz	uspto-grants-2016_09
ORD ID	ord-ef1975eaa436467cacd4ae20c0259985
Quellennotiz	uspto-grants-2016_09