5-Fluoro-3-methylbenzo[b]thiophene-2-sulphonyl chloride → HCID 178432000, Verbindung

Beteiligte Stoffe

Reaktionsschritte

The product was prepared according to General Procedure 1, described in Example 1, starting from 5-fluoro-3-methylbenzothiophene-2-sulfonyl chloride (Intermediate 14) (26 mg, 0.10 mmol) and 5-(3-amino-phenyl)tetrazole (31 mg, 0.19 mmol). The title compound was obtained in 36% yield (13.9 mg). MS (ESI+) calcd for C16H12FN5O2S2 389.041644, found 389.042334.

Herkunft & Nachweise