HuagongsheHuagongshe Chemie-Druckbericht · Nur für Forschungszwecke
Benzo[b]thiophene-3-boronic acid pinacol ester → (5-Benzo[b]thiophen-3-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-yl)-(4-morpholin-4-ylphenyl)amine
Beteiligte Stoffe
| Rolle | Name | HCID | Einwaage |
|---|---|---|---|
| Edukt | Benzo[b]thiophene-3-boronic acid pinacol ester | HCID 10658979 | — |
| Edukt | (5-Bromo-[1,2,4]triazolo[1,5-a]pyrazin-8-yl)-(4-morpholin-4-ylphenyl)amine | HCID 57589931 | — |
| Produkt | (5-Benzo[b]thiophen-3-yl-[1,2,4]triazolo[1,5-a]pyrazin-8-yl)-(4-morpholin-4-ylphenyl)amine | HCID 24888779 | — |
Reaktionsschritte
This compound may be prepared using methods as described for Compound 120, using (5-bromo-[1,2,4]triazolo[1,5-a]pyrazin-8-yl)-(4-morpholin-4-ylphenyl)amine and 4,4,5,5-tetramethyl-2-benzo[b]thiophen-3-yl-[1,3,2]dioxaborolane in step 4. LCMS: Rt 0.84 min (95%), m/z (ESI) 402 (M+H)+.
Herkunft & Nachweise
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patentnummer | US07915256B2 |
| Quelldatensatz | uspto-grants-2011_03 |
| ORD ID | ord-8e1c0897cf7543eb90b8e8ffa52f2eac |
| Quellennotiz | uspto-grants-2011_03 |