I[C:2]1[CH:3]=[C:4]([C:10]#[N:11])[C:5](=[CH:8][CH:9]=1)[C:6]#[N:7].[BH:12]([OH:14])[OH:13]>>[C:10]([C:4]1[CH:3]=[C:2]([B:12]([OH:14])[OH:13])[CH:9]=[CH:8][C:5]=1[C:6]#[N:7])#[N:11]The title compound was prepared according to Preparation 102 using 4-iodophthalonitrile to provide a mixture of the boronic acid and boronic ester. The mixture was taken on to the next step as crude.
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