Methyl 4-aminobenzoate → 4-(((Propan-2-yl)carbamoyl)amino)benzoic acid
Reaction equation
[CH:1]([NH:4][C:5](=[O:16])[NH:6][C:7]1C=C(C=CN=1)C(O)=O)([CH3:3])[CH3:2].N[C:18]1[CH:19]=[C:20]([CH:26]=[CH:27]N=1)[C:21]([O:23]CC)=[O:22].NC1C=CC(C(OC)=O)=CC=1>>[CH:1]([NH:4][C:5](=[O:16])[NH:6][C:7]1[CH:18]=[CH:19][C:20]([C:21]([OH:23])=[O:22])=[CH:26][CH:27]=1)([CH3:3])[CH3:2]Participants
4
Procedure
This compound is prepared analogously to Intermediate Y by replacing ethyl 2-aminoisonicotinate in step 1 with methyl 4-aminobenzoate; [M+H]+ 237.
Sources & evidence
- ORD record
- ord-c9d83fa7741e49488ee6d50850f19282
- Source dataset
- uspto-grants-2011_10
- Patent number
- US08039472B2
Reaction notes
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