(5-Cyano-2-Methoxyphenyl)Boronic Acid → HCID 86607716, compound

HRID 1752903

Reaction equation

HRID 1752903 reaction equation
Br[C:2]1[CH:3]=[C:4]([S:12]([NH2:15])(=[O:14])=[O:13])[CH:5]=[C:6]([CH:10]=[O:11])[C:7]=1[O:8][CH3:9].[C:16]([C:18]1[CH:19]=[CH:20][C:21]([O:27][CH3:28])=[C:22](B(O)O)[CH:23]=1)#[N:17]>>[C:16]([C:18]1[CH:19]=[CH:20][C:21]([O:27][CH3:28])=[C:22]([C:2]2[C:7]([O:8][CH3:9])=[C:6]([CH:10]=[O:11])[CH:5]=[C:4]([S:12]([NH2:15])(=[O:14])=[O:13])[CH:3]=2)[CH:23]=1)#[N:17]

Participants

3

Reactant 2

HCID 23005336(5-Cyano-2-Methoxyphenyl)Boronic AcidHCID 866076983-Bromo-5-formyl-4-methoxy-benzenesulfonamide

Product 1

HCID 86607716HCID 86607716, compound

Procedure

Proceeding as in Reference 19, but substituting 3-bromo-5-formyl-4-methoxy-benzenesulfonamide and 5-cyano-2-methoxy-benzeneboronic acid, gave 5′-cyano-5-formyl-6,2′-dimethoxybiphenyl-3-sulfonamide.

Sources & evidence

ORD record
ord-b79db7dcda3c445baa76cd6ef87c0a5c
Source dataset
uspto-grants-2015_10
Patent number
US09162986B2

Linked notes

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