1H-Indazole → (4-Chloro-phenyl)-(6-indazol-1-yl-pyrazin-2-yl)-amine
Reaction equation
C(OC(=O)[N:7]([C:15]1[CH:20]=[CH:19][C:18]([Cl:21])=[CH:17][CH:16]=1)[C:8]1[CH:13]=[N:12][CH:11]=[C:10](Cl)[N:9]=1)(C)(C)C.[NH:23]1[C:31]2[C:26](=[CH:27][CH:28]=[CH:29][CH:30]=2)[CH:25]=[N:24]1>>[Cl:21][C:18]1[CH:17]=[CH:16][C:15]([NH:7][C:8]2[CH:13]=[N:12][CH:11]=[C:10]([N:23]3[C:31]4[C:26](=[CH:27][CH:28]=[CH:29][CH:30]=4)[CH:25]=[N:24]3)[N:9]=2)=[CH:20][CH:19]=1Participants
3
Procedure
Were prepared according to Example 3 from (4-chloro-phenyl)-(6-chloro-pyrazin-2-yl)-carbamic acid tert-butyl ester and indazole.
Workup
- customWere prepared
Sources & evidence
- ORD record
- ord-b56cd66c0165466e8bb638068855aae1
- Source dataset
- uspto-grants-2013_04
- Patent number
- US08415358B2
Reaction notes
Loading…