5-Phenyl-1,3-oxazole-4-carboxylic acid → 5-Phenyl-oxazole-4-carboxylic acid [2-(5-methanesulfonyl-furan-2-ylmethyl)-2H-[1,2,3]triazol-4-yl]-amide

HRID 42916

Reaction equation

HRID 42916 reaction equation
[CH3:1][S:2]([C:5]1[O:9][C:8]([CH2:10][N:11]2[N:15]=[C:14]([NH2:16])[CH:13]=[N:12]2)=[CH:7][CH:6]=1)(=[O:4])=[O:3].[C:17]1([C:23]2[O:27][CH:26]=[N:25][C:24]=2[C:28](O)=[O:29])[CH:22]=[CH:21][CH:20]=[CH:19][CH:18]=1>>[CH3:1][S:2]([C:5]1[O:9][C:8]([CH2:10][N:11]2[N:15]=[C:14]([NH:16][C:28]([C:24]3[N:25]=[CH:26][O:27][C:23]=3[C:17]3[CH:18]=[CH:19][CH:20]=[CH:21][CH:22]=3)=[O:29])[CH:13]=[N:12]2)=[CH:7][CH:6]=1)(=[O:4])=[O:3]

Participants

3

Reactant 2

HCID 27762995-Phenyl-1,3-oxazole-4-carboxylic acidHCID 673652402-(5-Methanesulfonyl-furan-2-ylmethyl)-2H-[1,2,3]triazol-4-ylamine

Product 1

HCID 426465225-Phenyl-oxazole-4-carboxylic acid [2-(5-methanesulfonyl-furan-2-ylmethyl)-2H-[1,2,3]triazol-4-yl]-amide

Procedure

Following general procedure A, starting from 2-(5-methanesulfonyl-furan-2-ylmethyl)-2H-[1,2,3]triazol-4-ylamine and 5-phenyl-oxazole-4-carboxylic acid.

Sources & evidence

ORD record
ord-b53a1aeb98164a4488615638dbad658d
Source dataset
uspto-grants-2013_09
Patent number
US08536209B2

Linked notes

Loading…