3-Ethynylpyridine → HCID 58215581, compound

HRID 593568

Reaction equation

[C:1]([C:3]1[CH:4]=[N:5][CH:6]=[CH:7][CH:8]=1)#[CH:2].[F:9][C:10]1[CH:11]=[C:12]([C:14](I)=[CH:15][CH:16]=1)[NH2:13]>>[F:9][C:10]1[CH:11]=[C:12]2[C:14]([CH:2]=[C:1]([C:3]3[CH:4]=[N:5][CH:6]=[CH:7][CH:8]=3)[NH:13]2)=[CH:15][CH:16]=1

Participants

Reactant 2

HCID 1860033-Ethynylpyridine

HCID 27745125-Fluoro-2-iodoaniline

Product 1

HCID 58215581HCID 58215581, compound

Procedure

3-Ethynylpyridine and 3-fluoro-6-iodoaniline are processed according to the method described in Example 86 to give 6-fluoro-2-pyridin-3-yl-1H-indole. MS (ESI) m/z 213.0 (M+H)+.

Sources & evidence

ORD record: ord-49e3a277c10e4ee88174ac06dd5358a1
Source dataset: uspto-grants-2016_01
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US09242963B2

Linked notes

Loading…