3-Fluoro-2-iodobenzoic acid → 3-Fluoro-2-(2H-1,2,3-triazol-2-yl)benzoic acid

HRID 61218

Reaction equation

HRID 61218 reaction equation
C[C:2]1[CH:3]=[CH:4][C:5]([N:11]2[N:15]=[CH:14][CH:13]=[N:12]2)=[C:6]([CH:10]=1)[C:7]([OH:9])=[O:8].[F:16]C1C(I)=C(C=CC=1)C(O)=O.N1C=CN=N1>>[F:16][C:4]1[C:5]([N:11]2[N:15]=[CH:14][CH:13]=[N:12]2)=[C:6]([CH:10]=[CH:2][CH:3]=1)[C:7]([OH:9])=[O:8]

Participants

4

Reactant 3

HCID 223203083-Fluoro-2-iodobenzoic acidHCID 532601655-methyl-2-(2H-1,2,3-triazol-2-yl)benzoic acidHCID 178418936HCID 178418936, compound

Product 1

HCID 670865493-Fluoro-2-(2H-1,2,3-triazol-2-yl)benzoic acid

Procedure

The title compound was prepared following the same general protocol as described for 5-methyl-2-(2H-1,2,3-triazol-2-yl)benzoic acid in Example A11 using 3-fluoro-2-iodobenzoic acid and 1,2,3-triazole. ESI-MS (m/z): 208 [M+1]+.

Sources & evidence

ORD record
ord-2180607ac67546769ba6261ffde5e9a6
Source dataset
uspto-grants-2016_09
Patent number
US09440982B2

Linked notes

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