2-Fluoro-6-iodobenzoic acid → 2-Fluoro-6-(2H-1,2,3-triazol-2-yl)benzoic acid

HRID 61224

Reaction equation

HRID 61224 reaction equation
C[C:2]1[CH:3]=[CH:4][C:5]([N:11]2[N:15]=[CH:14][CH:13]=[N:12]2)=[C:6]([CH:10]=1)[C:7]([OH:9])=[O:8].[F:16]C1C=CC=C(I)C=1C(O)=O.N1C=CN=N1>>[F:16][C:10]1[CH:2]=[CH:3][CH:4]=[C:5]([N:11]2[N:15]=[CH:14][CH:13]=[N:12]2)[C:6]=1[C:7]([OH:9])=[O:8]

Participants

4

Procedure

The title compound was prepared following the same general protocol as described for 5-methyl-2-(2H-1,2,3-triazol-2-yl)benzoic acid in Example A11 using 2-fluoro-6-iodobenzoic acid and 1,2,3-triazole. ESI-MS (m/z): 208 [M+1]+.

Sources & evidence

ORD record
ord-90f6d143ac6f492fbd52cb87efa547d1
Source dataset
uspto-grants-2016_09
Patent number
US09440982B2

Linked notes

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