Reaction equation
[CH:1]1[CH:6]=[CH:5][C:4]([C:7]2[CH:12]=[CH:11][C:10]([CH2:13][CH2:14][NH2:15])=[CH:9][CH:8]=2)=[CH:3][CH:2]=1.ClC(OC1C=CC(F)=CC=1)=O.Cl[C:28]([O:30][C:31]1[CH:36]=[CH:35][C:34]([CH3:37])=[CH:33][CH:32]=1)=[O:29]>>[C:7]1([C:4]2[CH:3]=[CH:2][CH:1]=[CH:6][CH:5]=2)[CH:8]=[CH:9][C:10]([CH2:13][CH2:14][NH:15][C:28](=[O:29])[O:30][C:31]2[CH:36]=[CH:35][C:34]([CH3:37])=[CH:33][CH:32]=2)=[CH:11][CH:12]=1Participants
4
Procedure
The procedure is carried out in a manner similar to Example 4, replacing the 4-phenylbenzylamine with 2-(4-biphenyl)ethylamine and the 4-fluorophenyl chloroformate with 4-methylphenyl chloroformate.
Sources & evidence
- ORD record
- ord-267b9bc3419b43f0b93d351d986fb456
- Source dataset
- uspto-grants-2010_04
- Patent number
- US07696374B2
Linked notes
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