4-Methoxycarbonylphenylboronic acid → HCID 59264664, compound

Reaction equation

Br[C:2]1[N:3]=[C:4]([S:7][CH3:8])[S:5][CH:6]=1.[CH3:9][O:10][C:11]([C:13]1[CH:18]=[CH:17][C:16](B(O)O)=[CH:15][CH:14]=1)=[O:12]>>[CH3:9][O:10][C:11](=[O:12])[C:13]1[CH:18]=[CH:17][C:16]([C:2]2[N:3]=[C:4]([S:7][CH3:8])[S:5][CH:6]=2)=[CH:15][CH:14]=1

Participants

Reactant 2

HCID 27343694-Methoxycarbonylphenylboronic acid

HCID 164270944-Bromo-2-(methylthio)-1,3-thiazole

Product 1

HCID 59264664HCID 59264664, compound

Procedure

The title compound is prepared in a manner substantially analogous to Procedure M starting from 4-Bromo-2-methylsulfanyl-thiazole (CAS 204513-62-2) and 4-methoxycarbonylphenylboronic acid. MS (ES+) 266.2.

Sources & evidence

ORD record: ord-29d7a15600ac45f6adbb4d4d90df6066
Source dataset: uspto-grants-2010_04
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US07705025B2

Reaction notes

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