4-Bromo-2-methylbenzenesulfonyl chloride → 4-Bromo-2-methyl-N-((1-methyl-1H-indazol-5-yl)methyl)benzenesulfonamide
Reaction equation
[Br:1][C:2]1[CH:7]=[CH:6][C:5]([S:8](Cl)(=[O:10])=[O:9])=[C:4]([CH3:12])[CH:3]=1.[CH3:13][N:14]1[C:22]2[C:17](=[CH:18][C:19]([CH2:23][NH2:24])=[CH:20][CH:21]=2)[CH:16]=[N:15]1>>[Br:1][C:2]1[CH:7]=[CH:6][C:5]([S:8]([NH:24][CH2:23][C:19]2[CH:18]=[C:17]3[C:22](=[CH:21][CH:20]=2)[N:14]([CH3:13])[N:15]=[CH:16]3)(=[O:10])=[O:9])=[C:4]([CH3:12])[CH:3]=1Participants
3
Procedure
The titled compound was prepared according to the procedure described in step-1 of Example 1 from 4-bromo-2-methylbenzene-1-sulfonyl chloride and (1-methyl-1H-indazol-5-yl)methanamine.
Sources & evidence
- ORD record
- ord-51bf8aacdc73483c86e76e3c45c98b44
- Source dataset
- uspto-grants-2014_09
- Patent number