Ethyl 2-(hydroxyamino)benzoate → Ethyl 2-(((2-(trifluoromethyl)thiazol-4-yl)methoxy)amino)benzoate
反応式
[OH:1][NH:2][C:3]1[CH:13]=[CH:12][CH:11]=[CH:10][C:4]=1[C:5]([O:7][CH2:8][CH3:9])=[O:6].Br[CH2:15][C:16]1[N:17]=[C:18]([C:21]([F:24])([F:23])[F:22])[S:19][CH:20]=1>>[F:22][C:21]([F:24])([F:23])[C:18]1[S:19][CH:20]=[C:16]([CH2:15][O:1][NH:2][C:3]2[CH:13]=[CH:12][CH:11]=[CH:10][C:4]=2[C:5]([O:7][CH2:8][CH3:9])=[O:6])[N:17]=1参加物
3
実験手順
The titled compound was prepared using similar procedure as that of Example-1 (step-2) using ethyl 2-(hydroxyamino)benzoate and product of step 3 described above in 52% yield.
出典と根拠
- ORDレコード
- ord-3c9f90db63f14355ab673b252a23c5b1
- 出典データセット
- uspto-grants-2016_07
- 特許番号
- US09394300B2
反応ノート
読み込み中…