HCID 83702359、化合物 → HCID 89699660、化合物

HRID 1055740ノート

反応式

HRID 1055740 の反応式
[CH3:1][C:2]1[CH:8]=[CH:7][C:5]([NH2:6])=[CH:4][C:3]=1[N:9]1[C:16]2[N:12]([N:13]=[C:14]([C:17]3[CH:18]=[N:19][CH:20]=[CH:21][CH:22]=3)[CH:15]=2)[CH:11]=[CH:10]1.[C:23]([C:27]1[CH:28]=[C:29]([CH:33]=[C:34]([NH:36][CH3:37])[N:35]=1)[C:30](O)=[O:31])([CH3:26])([CH3:25])[CH3:24]>>[C:23]([C:27]1[CH:28]=[C:29]([CH:33]=[C:34]([NH:36][CH3:37])[N:35]=1)[C:30]([NH:6][C:5]1[CH:7]=[CH:8][C:2]([CH3:1])=[C:3]([N:9]2[C:16]3[N:12]([N:13]=[C:14]([C:17]4[CH:18]=[N:19][CH:20]=[CH:21][CH:22]=4)[CH:15]=3)[CH:11]=[CH:10]2)[CH:4]=1)=[O:31])([CH3:26])([CH3:24])[CH3:25]

参加物

3

反応物 2

HCID 83702359HCID 83702359、化合物HCID 897000234-Methyl-3-[6-(pyridin-3-yl)-1H-imidazo[1,2-b]pyrazol-1-yl]aniline

生成物 1

HCID 89699660HCID 89699660、化合物

実験手順

60 mg (0.21 mmol) of the compound of Example 6A and 43 mg (0.21 mmol) of the compound of Example 44A were reacted analogously to the procedure of Example 33, except that in this case the reaction time was 16 h. This gave 31 mg (31% of theory) of the title compound.

出典と根拠

ORDレコード
ord-c5928560833f44658e84f44c806a5b1d
出典データセット
uspto-grants-2016_07
特許番号
US09394309B2

反応ノート

読み込み中…