Cyclopropylamine → 2-Cyclopropylamino-5-sulfamoylbenzoic acid

反応式

F[C:2]1[CH:10]=[CH:9][C:8]([S:11](=[O:14])(=[O:13])[NH2:12])=[CH:7][C:3]=1[C:4]([OH:6])=[O:5].[CH:15]1([NH2:18])[CH2:17][CH2:16]1>>[CH:15]1([NH:18][C:2]2[CH:10]=[CH:9][C:8]([S:11](=[O:14])(=[O:13])[NH2:12])=[CH:7][C:3]=2[C:4]([OH:6])=[O:5])[CH2:17][CH2:16]1

参加物

反応物 2

HCID 69828Cyclopropylamine

HCID 24926842-Fluoro-5-sulfamoylbenzoic acid

生成物 1

HCID 198486222-Cyclopropylamino-5-sulfamoylbenzoic acid

実験手順

The title compound is prepared from 2-fluoro-5-sulfamoylbenzoic acid and cyclopropylamine in substantially the same manner as in Reference Example 87.

出典と根拠

ORDレコード: ord-69ac9c265e054a42a6ec193baf2627f7
出典データセット: uspto-grants-1989_09
DOI: 10.6084/m9.figshare.5104873.v1
特許番号: US04870074

反応ノート

読み込み中…