3-(7-Fluoro-2-quinolinylmethoxy)aniline → 4-[3-(7-Fluoro-2-quinolinylmethoxy)phenylamino]-2,2-dipropyl-4-oxobutanoic acid
反応式
[CH2:1]([C:4]1([CH2:11][CH2:12][CH3:13])[CH2:9][C:8](=[O:10])[O:7][C:5]1=[O:6])[CH2:2][CH3:3].[F:14][C:15]1[CH:24]=[C:23]2[C:18]([CH:19]=[CH:20][C:21]([CH2:25][O:26][C:27]3[CH:28]=[C:29]([CH:31]=[CH:32][CH:33]=3)[NH2:30])=[N:22]2)=[CH:17][CH:16]=1>>[F:14][C:15]1[CH:24]=[C:23]2[C:18]([CH:19]=[CH:20][C:21]([CH2:25][O:26][C:27]3[CH:28]=[C:29]([NH:30][C:8](=[O:10])[CH2:9][C:4]([CH2:11][CH2:12][CH3:13])([CH2:1][CH2:2][CH3:3])[C:5]([OH:7])=[O:6])[CH:31]=[CH:32][CH:33]=3)=[N:22]2)=[CH:17][CH:16]=1参加物
3
実験手順
The title compound is prepared analogously to the compound described in Example 20 from 2,2-dipropylsuccinic acid anhydride and 3-(7-fluoro-2-quinolinylmethoxy)aniline; beige crystals of m.p. 155°-156°.
出典と根拠
- ORDレコード
- ord-5c6d46f301524830b20db1cdafe21037
- 出典データセット
- uspto-grants-1996_04
- 特許番号
- US05508408
反応ノート
読み込み中…