化工社化工社 化学情報印刷レポート · 研究参考用
3-(N,N-Dimethylsulphonamido)benzeneboronic acid → 3-(2-{[dihydroxy(1-methylethyl)-lambda4-sulfanyl]amino}-2,3-dihydro-1H-inden-5-yl)-N,N-dimethylbenzenesulfonamide
関与物質
| 役割 | 名称 | HCID | 仕込み量 |
|---|---|---|---|
| 反応物 | 3-(N,N-Dimethylsulphonamido)benzeneboronic acid | HCID 44119634 | — |
| 反応物 | N-(5-iodo-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamide | HCID 46899809 | — |
| 生成物 | 3-(2-{[dihydroxy(1-methylethyl)-lambda4-sulfanyl]amino}-2,3-dihydro-1H-inden-5-yl)-N,N-dimethylbenzenesulfonamide | HCID 68447569 | — |
反応手順
The title compound was prepared from N-(5-iodo-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamide and {3-[(dimethylamino)sulfonyl]phenyl}boronic acid (WO2003004472) in a similar manner to Example 1.
情報源と証拠
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| 特許番号 | US07741351B2 |
| 出典データセット | uspto-grants-2010_06 |
| ORD ID | ord-42b9c346e4594c3b87f17142402350a2 |
| 出典メモ | uspto-grants-2010_06 |