Ethyl 3-{[(4-aminophenyl)carbonyl](methyl)amino}propanoate → HCID 66777908、化合物
反応式
[CH:1]1([CH:7]([C:9]2[N:10]=[C:11]3[CH:16]=[CH:15][C:14]([C:17]([F:20])([F:19])[F:18])=[CH:13][N:12]3[CH:21]=2)O)[CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1.[NH2:22][C:23]1[CH:28]=[CH:27][C:26]([C:29]([N:31]([CH3:39])[CH2:32][CH2:33][C:34]([O:36]CC)=[O:35])=[O:30])=[CH:25][CH:24]=1>>[CH:1]1([CH:7]([NH:22][C:23]2[CH:24]=[CH:25][C:26]([C:29]([N:31]([CH3:39])[CH2:32][CH2:33][C:34]([OH:36])=[O:35])=[O:30])=[CH:27][CH:28]=2)[C:9]2[N:10]=[C:11]3[CH:16]=[CH:15][C:14]([C:17]([F:20])([F:19])[F:18])=[CH:13][N:12]3[CH:21]=2)[CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1参加物
3
実験手順
Using cyclohexyl[6-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]methanol (1.1 g) synthesized above and ethyl 3-{[(4-aminophenyl)carbonyl](methyl)amino}propanoate (0.94 g) synthesized in Example 2(2) and in the same manner as in Example 4, the title object compound (3.0 mg, 2%) was obtained as an oil.
出典と根拠
- ORDレコード
- ord-86004a69583b45d4851af958a5940d37
- 出典データセット
- uspto-grants-2013_05