Ethylamine → N-[4-(1-Aminoethyl)-2-methoxyphenyl]methanesulfonamide
反応式
[CH3:1][O:2][C:3]1[CH:4]=[C:5]([CH:14]([NH:16]C(=O)OCC2C=CC=CC=2)[CH3:15])[CH:6]=[CH:7][C:8]=1[NH:9][S:10]([CH3:13])(=[O:12])=[O:11].C(N)C>>[CH3:1][O:2][C:3]1[CH:4]=[C:5]([CH:14]([NH2:16])[CH3:15])[CH:6]=[CH:7][C:8]=1[NH:9][S:10]([CH3:13])(=[O:12])=[O:11]参加物
3
実験手順
Through similar procedure to that in Example 1-2 excepting using Benzyl N-{1-[3-methoxy-4-(methylsulfonylamino)phenyl]ethyl}carbamate (14-1) as a starting material, □1□3-Methoxy-4-(methylsulfonylamino)phenyl]ethyl amine (14-3, CHK-570) having following physicochemical properties was synthesized:
後処理
- customwas synthesized
出典と根拠
- ORDレコード
- ord-8d2a44d3740347898bf963d84966a48b
- 出典データセット
- uspto-grants-2014_02
- 特許番号
- US08642657B2
反応ノート
読み込み中…