戻る
化工社化工社 化学情報印刷レポート · 研究参考用
HRID 351000作成日：2026年10月26日

(+/-)-2-[4-({[2-(Benzo[2,1,3]oxadiazol-5-yloxy)-pyridine-3-carbonyl]-amino}-methyl)-3-fluoro-phenoxy]-propionic acid tert-butyl ester → (+/-)-2-[4-({[2-(Benzo[2,1,3]thiadiazol-5-yloxy)-pyridine-3-carbonyl]-amino}-methyl)-3-fluoro-phenoxy]-propionic acid

https://huagongshe.com/reaction/351000

反応式

関与物質

役割名称HCID仕込み量
反応物(+/-)-2-[4-({[2-(Benzo[2,1,3]oxadiazol-5-yloxy)-pyridine-3-carbonyl]-amino}-methyl)-3-fluoro-phenoxy]-propionic acid tert-butyl esterHCID 23529359—
反応物(+)-2-[4-({[2-(Benzo[2,1,3]thiadiazol-5-yloxy)-pyridine-3-carbonyl]-amino}-methyl)-3-fluoro-phenoxy]-propionic acid tert-butyl esterHCID 23529360—
生成物(+/-)-2-[4-({[2-(Benzo[2,1,3]thiadiazol-5-yloxy)-pyridine-3-carbonyl]-amino}-methyl)-3-fluoro-phenoxy]-propionic acidHCID 10115978—

反応手順

The compound of Formula (5.5.7) was prepared in a manner analogous to that described in Example 3, substituting (+)-2-[4-({[2-(benzo[2,1,3]thiadiazol-5-yloxy)-pyridine-3-carbonyl]-amino}-methyl)-3-fluoro-phenoxy]-propionic acid tert-butyl ester for the corresponding (±)-2-[4-({[2-(benzo[2,1,3]oxadiazol-5-yloxy)-pyridine-3-carbonyl]-amino}-methyl)-3-fluoro -phenoxy]-propionic acid tert-butyl ester material.

情報源と証拠

DOI10.6084/m9.figshare.5104873.v1
特許番号US07183293B2
出典データセットuspto-grants-2007_02
ORD IDord-fe38f03f16fd4063a98056ba93afe392
出典メモuspto-grants-2007_02