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3-(2,6-Dichlorobenzyloxy)-5-bromopyridin-2-amine → ethyl 5-{6-amino-5-[(2,6-dichlorobenzyl)oxy]pyridin-3-yl}-1H-indole-2-carboxylate
関与物質
| 役割 | 名称 | HCID | 仕込み量 |
|---|---|---|---|
| 反応物 | 3-(2,6-Dichlorobenzyloxy)-5-bromopyridin-2-amine | HCID 21111487 | — |
| 反応物 | Ethyl 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole-2-carboxylate | HCID 21111505 | — |
| 生成物 | ethyl 5-{6-amino-5-[(2,6-dichlorobenzyl)oxy]pyridin-3-yl}-1H-indole-2-carboxylate | HCID 10253528 | — |
反応手順
5-[6-Amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-1H-indole-2-carboxylic acid ethyl ester was prepared from 5-bromo-3-(2,6-dichloro-benzyloxy)-pyridin-2-ylamine and 5-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-1H-indole-2-carboxylic acid ethyl ester following procedure 3.
情報源と証拠
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| 特許番号 | US08106197B2 |
| 出典データセット | uspto-grants-2012_01 |
| ORD ID | ord-26233665d8404da7a137131f63bb652a |
| 出典メモ | uspto-grants-2012_01 |