化工社化工社 化学情報印刷レポート · 研究参考用
5-Bromo-[1,2,4]triazolo[1,5-a]pyridin-2-amine → 5-[4-[(1,1-Dioxo-1,4-thiazinan-4-yl)methyl]phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine
関与物質
| 役割 | 名称 | HCID | 仕込み量 |
|---|---|---|---|
| 反応物 | 5-Bromo-[1,2,4]triazolo[1,5-a]pyridin-2-amine | HCID 25215939 | — |
| 反応物 | (4-((1,1-Dioxidothiomorpholino)methyl)phenyl)boronic acid | HCID 54970580 | — |
| 生成物 | 5-[4-[(1,1-Dioxo-1,4-thiazinan-4-yl)methyl]phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine | HCID 67479440 | — |
反応手順
5-{-4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-amine was prepared from 5-bromo-[1,2,4]triazolo[1,5-a]pyridin-2-ylamine and 4-[(4-boronophenyl)methyl]-thiomorpholine 1,1-dioxide in a manner analogous to Step 2c. The reaction product was taken on to the next step.
情報源と証拠
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| 特許番号 | US08633173B2 |
| 出典データセット | uspto-grants-2014_01 |
| ORD ID | ord-042a536bb51f4d9ca93476251e8038f5 |
| 出典メモ | uspto-grants-2014_01 |