3-[(E)-2-(4-chlorophenyl)vinyl]-4-methoxy-benzoic acid → 3-[(E)-2-(4-chlorophenyl)-vinyl]-4-methoxy-N-((2S,3S)-2,3,4-trihydroxy-butyl)benzamide
反応式
[Cl:1][C:2]1[CH:7]=[CH:6][C:5](/[CH:8]=[CH:9]/[C:10]2[CH:11]=[C:12]([CH:16]=[CH:17][C:18]=2[O:19][CH3:20])[C:13]([OH:15])=O)=[CH:4][CH:3]=1.[NH2:21][CH2:22][C@H:23]([OH:28])[C@@H:24]([OH:27])[CH2:25][OH:26]>>[Cl:1][C:2]1[CH:3]=[CH:4][C:5](/[CH:8]=[CH:9]/[C:10]2[CH:11]=[C:12]([CH:16]=[CH:17][C:18]=2[O:19][CH3:20])[C:13]([NH:21][CH2:22][C@H:23]([OH:28])[C@@H:24]([OH:27])[CH2:25][OH:26])=[O:15])=[CH:6][CH:7]=1参加物
3
実験手順
The captioned compound was synthesized from 4-methoxy-3-[(E)-2-(4-chlorophenyl)vinyl]benzoic acid obtained in step B of Example 2-2-7 and (2S,3S)-4-amino-1,2,3-butanetriol (CAS registry number: 168113-19-7) in accordance with the same procedure as in the methods described in step C of Example 1-2-3.
出典と根拠
- ORDレコード
- ord-c0b8e3bdf8e64fde93bf4ad5282ce0a9
- 出典データセット
- uspto-grants-2010_04
- 特許番号
- US07705053B2
反応ノート
読み込み中…