1-Benzylazetidine-2-carboxylic acid → HCID 71186307、化合物
反応式
[CH2:1]([N:8]1[CH2:11][CH2:10][CH:9]1[C:12]([OH:14])=O)[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.Cl.[NH2:16][C@H:17]([C:19]1[CH:28]=[CH:27][C:22]([C:23]([O:25][CH3:26])=[O:24])=[CH:21][CH:20]=1)[CH3:18]>>[CH2:1]([N:8]1[CH2:11][CH2:10][CH:9]1[C:12]([NH:16][C@H:17]([C:19]1[CH:28]=[CH:27][C:22]([C:23]([O:25][CH3:26])=[O:24])=[CH:21][CH:20]=1)[CH3:18])=[O:14])[C:2]1[CH:3]=[CH:4][CH:5]=[CH:6][CH:7]=1参加物
3
実験手順
The title compound (D76) (98 mg) was prepared according to the general procedure for amides preparation (Method C) starting from 1-benzylazetidine-2-carboxylic acid (100 mg, available from Apollo#OR7040) and (S)-methyl 4-(1-aminoethyl)benzoate hydrochloride (113 mg). Reaction time: 1 h
後処理
- customReaction time
- custom1 h
出典と根拠
- ORDレコード
- ord-83f076cccdb742349530cc10143933be