化工社化工社 化学情報印刷レポート · 研究参考用
3-Fluorophenol → 1-Benzhydryl-3-(3-fluorophenoxy)azetidine
関与物質
| 役割 | 名称 | HCID | 仕込み量 |
|---|---|---|---|
| 反応物 | 3-Fluorophenol | HCID 9743 | — |
| 反応物 | 1-(Diphenylmethyl)azetidin-3-yl methanesulfonate | HCID 2758716 | — |
| 生成物 | 1-Benzhydryl-3-(3-fluorophenoxy)azetidine | HCID 19799621 | 80.9% |
反応手順
The title compound (D22) (1.93 g) was prepared according to the experimental procedure described in Description 21 starting from 1-benzhydrylazetidin-3-yl methanesulfonate (D19) (2.5 g, 7.87 mmol) and 3-fluorophenol (0.642 ml, 7.16 mmol).
情報源と証拠
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| 特許番号 | US08828987B2 |
| 出典データセット | uspto-grants-2014_09 |
| ORD ID | ord-83dabc3e49b94d36991f1f54a4471d05 |
| 出典メモ | uspto-grants-2014_09 |