化工社化工社 化学情報印刷レポート · 研究参考用
3-Methyl-2-thenoic acid → 5-(3-methyl-2-thienoyl)amino-3-(1-methylpiperidin-4-yl)-1H-indole
関与物質
| 役割 | 名称 | HCID | 仕込み量 |
|---|---|---|---|
| 反応物 | 3-Methyl-2-thenoic acid | HCID 90269 | — |
| 反応物 | 3-(1-Methylpiperidin-4-yl)-1h-indol-5-amine | HCID 11831220 | — |
| 生成物 | 5-(3-methyl-2-thienoyl)amino-3-(1-methylpiperidin-4-yl)-1H-indole | HCID 22611475 | 90.5% |
反応手順
Beginning with 7.0 mg (0.03 mMol) 5-amino-3-(1-methylpiperidin-4-yl)-1H-indole and 12.8 mg (0.09 mMol) 3-methyl-2-thienoic acid, 9.6 mg (90%) of the title compound were recovered.
情報源と証拠
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| 特許番号 | US06380201B1 |
| 出典データセット | uspto-grants-2002_04 |
| ORD ID | ord-fcc1503bad3b4d5ab557ca9fec9ba627 |
| 出典メモ | uspto-grants-2002_04 |