Pyrazolo[1,5-a]pyriMidine-5-carbonitrile → Pyrazolo[1,5-a]pyrimidine-5-methanamine
反応式
[N:1]1[N:5]2[CH:6]=[CH:7][C:8]([C:10]#[N:11])=[N:9][C:4]2=[CH:3][CH:2]=1.S1C2=NC=CC=C2C(CN)=C1>>[N:1]1[N:5]2[CH:6]=[CH:7][C:8]([CH2:10][NH2:11])=[N:9][C:4]2=[CH:3][CH:2]=1参加物
3
実験手順
Intermediate M was prepared from pyrazolo[1,5-a]pyrimidine-5-carbonitrile (M−1) following similar procedures for synthesizing intermediate J from J-4, as described above. MS (m/z): 149 (M+1)+.
出典と根拠
- ORDレコード
- ord-cbbc6779e255437998c8fb9d672e3d26
- 出典データセット
- uspto-grants-2015_03
- 特許番号
- US08987269B2
反応ノート
読み込み中…