化工社化工社 化学情報印刷レポート · 研究参考用
(S)-2-methoxycarbonylamino-3,3-diphenyl-propionic acid → Ppl-100
関与物質
| 役割 | 名称 | HCID | 仕込み量 |
|---|---|---|---|
| 反応物 | (S)-2-methoxycarbonylamino-3,3-diphenyl-propionic acid | HCID 10017620 | — |
| 反応物 | (1S)-4-amino-N-(5-amino-1-hydroxymethyl-pentyl)-N-isobutyl-benzenesulfonamide | HCID 20595420 | — |
| 生成物 | Ppl-100 | HCID 513956 | — |
反応手順
The title compound was prepared from (1S)-4-amino-N-(5-amino-1-hydroxymethyl-pentyl)-N-isobutyl-benzenesulfonamide (XII) (example 28, step D) as described in general procedure B using (2S)-2-methoxycarbonylamino-3,3-diphenyl-propionic acid (step A). The final product was obtained in 67% yield (121 mg).
情報源と証拠
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| 特許番号 | US06632816B1 |
| 出典データセット | uspto-grants-2003_10 |
| ORD ID | ord-12c80c89f857458ab322c25173d56050 |
| 出典メモ | uspto-grants-2003_10 |