HCID 10539351, 화합물 → HCID 54361485, 화합물

HRID 1274988노트

반응식

HRID 1274988 반응식
[NH2:1][C:2]1[CH:3]=[C:4]2[C:9](=[CH:10][CH:11]=1)[CH2:8][CH:7]([CH2:12][C:13]([O:15][C:16]([CH3:19])([CH3:18])[CH3:17])=[O:14])[CH2:6][CH2:5]2.[N:20]1[CH:25]=[CH:24][CH:23]=[CH:22][C:21]=1[NH:26][CH2:27][CH2:28][C:29](O)=[O:30]>>[N:20]1[CH:25]=[CH:24][CH:23]=[CH:22][C:21]=1[NH:26][CH2:27][CH2:28][C:29]([NH:1][C:2]1[CH:3]=[C:4]2[C:9](=[CH:10][CH:11]=1)[CH2:8][CH:7]([CH2:12][C:13]([O:15][C:16]([CH3:19])([CH3:18])[CH3:17])=[O:14])[CH2:6][CH2:5]2)=[O:30]

참가 물질

3

반응물 2

HCID 10539351HCID 10539351, 화합물HCID 119834723-(pyridin-2-ylamino)propanoic Acid

생성물 1

HCID 54361485HCID 54361485, 화합물

실험 절차

Following the procedure of Example 32(a), except substituting tert-butyl (6-amino-tetralin-2-yl)acetate, Fisher, et. al., EO 0635492, Scheme 12 and Example 28, parts A-D, for the compound of Preparation O(d) and substituting N-(2-pyridinyl)-β-alanine, Chowdhary, et. al., Indian J. Chem., 1990, 29A, 280-284, for the compound of Preparation V, gives the title compound.

후처리

  1. customfor the compound of Preparation O(d)

출처 및 근거

ORD 기록
ord-5322ee7fced04f3d8f17b97218c50eff
출처 데이터셋
uspto-grants-2000_12
특허 번호
US06159964

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