3-Isoxazolamine → 1-(5-tert-Butyl-isoxazol-3-ylcarbamoyl)-propyl-carbamic acid tert-butyl ester

HRID 1294825

반응식

HRID 1294825 반응식
[C:1]([O:5][C:6](=[O:24])[NH:7][CH:8]([C:12](=[O:23])[NH:13][C:14]1[CH:18]=[C:17]([C:19]([CH3:22])([CH3:21])[CH3:20])[O:16][N:15]=1)[CH2:9][CH2:10]C)([CH3:4])([CH3:3])[CH3:2].NC1C=CON=1>>[C:1]([O:5][C:6](=[O:24])[NH:7][CH:8]([C:12](=[O:23])[NH:13][C:14]1[CH:18]=[C:17]([C:19]([CH3:22])([CH3:21])[CH3:20])[O:16][N:15]=1)[CH2:9][CH3:10])([CH3:3])([CH3:2])[CH3:4]

참가 물질

3

반응물 2

HCID 18102163-IsoxazolamineHCID 69419406[1-(5-Tert-butyl-isoxazol-3-ylcarbamoyl)butyl]-carbamic acid tert-butyl ester

생성물 1

HCID 694241221-(5-tert-Butyl-isoxazol-3-ylcarbamoyl)-propyl-carbamic acid tert-butyl ester

실험 절차

Prepared by the analogous method for the preparation of [1-(5-tert-butyl-isoxazol-3-ylcarbamoyl)butyl]-carbamic acid tert-butyl ester, starting with an appropriate amino-isoxazole (1 a-b) together with an appropriate N-t-BOC-amino acid methyl or ethyl ester.

출처 및 근거

ORD 기록
ord-d7f47e78ef3147b1bb761a63a2b37375
출처 데이터셋
uspto-grants-2007_07
특허 번호
US07241786B2

연결된 노트

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