Boronic Acid → Quinoxalin-6-ylboronic acid hydrochloride

HRID 1446111노트

반응식

HRID 1446111 반응식
Br[C:2]1[CH:3]=[C:4]2[C:9](=[CH:10][CH:11]=1)[N:8]=[CH:7][C:6]([N+:12]([O-])=O)=C2[Cl:15].NC1C=CC(C(CC)(CC)C#N)=CC=1.[BH:30]([OH:32])[OH:31]>>[ClH:15].[N:8]1[C:9]2[CH:10]=[CH:11][C:2]([B:30]([OH:32])[OH:31])=[CH:3][C:4]=2[N:12]=[CH:6][CH:7]=1

참가 물질

4

반응물 3

HCID 61668Boronic AcidHCID 138269352-(4-Amino-phenyl)-2-ethyl-butyronitrileHCID 219841286-Bromo-4-chloro-3-nitroquinoline

생성물 1

HCID 45073595Quinoxalin-6-ylboronic acid hydrochloride

실험 절차

The following compounds (Table 2) are prepared in a similar manner as described in Example 1 by reacting 6-bromo-4-chloro-3-nitro-quinoline (Example 1c) with 2-(4-amino-phenyl)-2-ethyl-butyronitrile (Example 12a), and with the appropriate boronic acid:

후처리

  1. customThe following compounds (Table 2) are prepared in a similar manner

출처 및 근거

ORD 기록
ord-4bcba08be1ea4c92b46c0eb2771eb530
출처 데이터셋
uspto-grants-2010_02
특허 번호
US07667039B2

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