3-Pyridinylboronic acid → 3-(1-Benzyl-2-methyl-6-pyridin-3-yl-1H-indol-3-ylsulfanyl)-benzoic acid methyl ester

HRID 1466775

반응식

HRID 1466775 반응식
[CH3:1][O:2][C:3](=[O:29])[C:4]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10][C:11]2[C:19]3[C:14](=[CH:15][C:16](Br)=[CH:17][CH:18]=3)[N:13]([CH2:21][C:22]3[CH:27]=[CH:26][CH:25]=[CH:24][CH:23]=3)[C:12]=2[CH3:28])[CH:5]=1.[N:30]1[CH:35]=[CH:34][CH:33]=[C:32](B(O)O)[CH:31]=1>>[CH3:1][O:2][C:3](=[O:29])[C:4]1[CH:9]=[CH:8][CH:7]=[C:6]([S:10][C:11]2[C:19]3[C:14](=[CH:15][C:16]([C:32]4[CH:31]=[N:30][CH:35]=[CH:34][CH:33]=4)=[CH:17][CH:18]=3)[N:13]([CH2:21][C:22]3[CH:27]=[CH:26][CH:25]=[CH:24][CH:23]=3)[C:12]=2[CH3:28])[CH:5]=1

참가 물질

3

반응물 2

HCID 27343783-Pyridinylboronic acidHCID 667652363-(1-Benzyl-6-bromo-2-methyl-1H-indol-3-ylsulfanyl)-benzoic acid methyl ester

생성물 1

HCID 667655523-(1-Benzyl-2-methyl-6-pyridin-3-yl-1H-indol-3-ylsulfanyl)-benzoic acid methyl ester

실험 절차

Prepared according to the procedure described in Example 11, Step 1, using the following starting materials: 3-(1-benzyl-6-bromo-2-methyl-1H-indol-3-ylsulfanyl)-benzoic acid methyl ester and 3-pyridineboronic acid.

후처리

  1. customPrepared

출처 및 근거

ORD 기록
ord-1a080162b7a84de28afa006ab012ba57
출처 데이터셋
uspto-grants-2015_04
특허 번호
US09000025B2

연결된 노트

불러오는 중…