Phenylboronic Acid → HCID 58398084, 화합물

반응식

Br[C:2]1[CH:7]=[CH:6][N:5]2[N:8]=[C:9]([NH:11][CH:12]3[CH2:17][CH2:16][N:15]([C:18]4[S:22][N:21]=[C:20]([CH3:23])[N:19]=4)[CH2:14][CH2:13]3)[N:10]=[C:4]2[CH:3]=1.[C:24]1(B(O)O)[CH:29]=[CH:28][CH:27]=[CH:26][CH:25]=1>>[CH3:23][C:20]1[N:19]=[C:18]([N:15]2[CH2:16][CH2:17][CH:12]([NH:11][C:9]3[N:10]=[C:4]4[CH:3]=[C:2]([C:24]5[CH:29]=[CH:28][CH:27]=[CH:26][CH:25]=5)[CH:7]=[CH:6][N:5]4[N:8]=3)[CH2:13][CH2:14]2)[S:22][N:21]=1

참가 물질

반응물 2

HCID 66827Phenylboronic Acid

HCID 67344430HCID 67344430, 화합물

생성물 1

HCID 58398084HCID 58398084, 화합물

실험 절차

Prepared in analogy to example 66c from (7-bromo-[1,2,4]triazolo[1,5-a]pyridin-2-yl)-[1-(3-methyl-[1,2,4]thiadiazol-5-yl)-piperidin-4-yl]-amine and phenyl boronic acid. The title compound was obtained as off-white foam.

출처 및 근거

ORD 기록: ord-a81f0542711441fcae4d5025f58c4ef7
출처 데이터셋: uspto-grants-2013_07
DOI: 10.6084/m9.figshare.5104873.v1
특허 번호: US08486967B2

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