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Huagongshe화공사 화학 정보 인쇄 보고서 · 연구 참고용
HRID 57840생성일: 2026년 10월 26일

1-Ethyl-1H-pyrazole-4-boronic acid, pinacol ester → N-(6-(6-(1-ethyl-1H-pyrazol-4-yl)-1H-pyrazolo[4,3-c]pyridin-1-yl)pyridin-2-yl)azepan-3-amine

https://huagongshe.com/reaction/57840

반응식

참여 물질

역할이름HCID투입량
반응물1-Ethyl-1H-pyrazole-4-boronic acid, pinacol esterHCID 11379045—
반응물tert-Butyl 3-aminoazepane-1-carboxylateHCID 23068067—
생성물N-(6-(6-(1-ethyl-1H-pyrazol-4-yl)-1H-pyrazolo[4,3-c]pyridin-1-yl)pyridin-2-yl)azepan-3-amineHCID 867070442.8%

반응 단계

Following the procedures as described in EXAMPLE 8 and starting with 1-ethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole and tert-butyl 3-aminoazepane-1-carboxylate, 143 was obtained as an off-white solid (3.6 mg, 2.8%) over 2 steps. MS (ESI) m/z: 403.2 [M+H]+

출처 및 근거

DOI10.6084/m9.figshare.5104873.v1
특허 번호US09434725B2
출처 데이터셋uspto-grants-2016_09
ORD IDord-dbdd60ba933d40efa4e90715a30d0c9e
출처 메모uspto-grants-2016_09