3-Methoxybenzenesulfonyl chloride → 3-[2-(4-m-Methoxybenzenesulphonamido-1-piperidyl)ethyl]indole

HRID 66306

반응식

HRID 66306 반응식
O.[NH2:2][CH:3]1[CH2:8][CH2:7][N:6]([CH2:9][CH2:10][C:11]2[C:19]3[C:14](=[CH:15][CH:16]=[CH:17][CH:18]=3)[NH:13][CH:12]=2)[CH2:5][CH2:4]1.[CH3:20][O:21][C:22]1[CH:23]=[C:24]([S:28](Cl)(=[O:30])=[O:29])[CH:25]=[CH:26][CH:27]=1>>[CH3:20][O:21][C:22]1[CH:23]=[C:24]([S:28]([NH:2][CH:3]2[CH2:8][CH2:7][N:6]([CH2:9][CH2:10][C:11]3[C:19]4[C:14](=[CH:15][CH:16]=[CH:17][CH:18]=4)[NH:13][CH:12]=3)[CH2:5][CH2:4]2)(=[O:30])=[O:29])[CH:25]=[CH:26][CH:27]=1

참가 물질

3

반응물 2

HCID 27375043-Methoxybenzenesulfonyl chlorideHCID 203843533-[2-(4-Aminopiperidyl)ethyl]indole, hydrate

생성물 1

HCID 227548393-[2-(4-m-Methoxybenzenesulphonamido-1-piperidyl)ethyl]indole

실험 절차

Using an analogous procedure to Example 1 3-[2-(4-amino-1-piperidyl)ethyl]indole monohydrate may be reacted with m-methoxybenzenesulphonyl chloride to give the title compound.

출처 및 근거

ORD 기록
ord-bd239b7bbe774ba9ab9b0916e1749cde
출처 데이터셋
uspto-grants-1978_12
특허 번호
US04131680

연결된 노트

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