3,4-Dichlorobenzeneboronic acid → HCID 86595309, compound

HRID 1009704Notes

Reaction equation

HRID 1009704 reaction equation
[Cl:1][C:2]1[CH:7]=[C:6]([C:8]#[C:9][C:10]2[N:11]=[C:12]([CH3:15])[NH:13][CH:14]=2)[CH:5]=[CH:4][N:3]=1.[Cl:16][C:17]1[CH:18]=[C:19](B(O)O)[CH:20]=[CH:21][C:22]=1[Cl:23]>>[Cl:1][C:2]1[CH:7]=[C:6]([C:8]#[C:9][C:10]2[N:11]=[C:12]([CH3:15])[N:13]([C:20]3[CH:19]=[CH:18][C:17]([Cl:16])=[C:22]([Cl:23])[CH:21]=3)[CH:14]=2)[CH:5]=[CH:4][N:3]=1

Participants

3

Reactant 2

HCID 27343303,4-Dichlorobenzeneboronic acidHCID 178418879HCID 178418879, compound

Product 1

HCID 86595309HCID 86595309, compound

Procedure

The title compound, MS: m/e=363.7 (M+H+), was prepared in accordance with the general method of example 7 from 2-chloro-4-(2-methyl-1H-imidazol-4-ylethynyl)-pyridine and 3,4-dichlorobenzene boronic acid.

Sources & evidence

ORD record
ord-085b122da9ff4db8827567c99f86706f
Source dataset
uspto-grants-2011_07
Patent number
US07973165B2

Reaction notes

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