3-Cyanophenylboronic acid → HCID 86595321, compound

HRID 1009720Notes

Reaction equation

HRID 1009720 reaction equation
[Cl:1][C:2]1[CH:7]=[C:6]([C:8]#[C:9][C:10]2[N:11]=[C:12]([CH3:15])[NH:13][CH:14]=2)[CH:5]=[CH:4][N:3]=1.[C:16]([C:18]1[CH:19]=[C:20](B(O)O)[CH:21]=[CH:22][CH:23]=1)#[N:17]>>[Cl:1][C:2]1[CH:7]=[C:6]([C:8]#[C:9][C:10]2[N:11]=[C:12]([CH3:15])[N:13]([C:22]3[CH:23]=[C:18]([CH:19]=[CH:20][CH:21]=3)[C:16]#[N:17])[CH:14]=2)[CH:5]=[CH:4][N:3]=1

Participants

3

Reactant 2

HCID 27343253-Cyanophenylboronic acidHCID 178418879HCID 178418879, compound

Product 1

HCID 86595321HCID 86595321, compound

Procedure

The title compound, MS: m/e=319.8 (M+H+), was prepared in accordance with the general method of example 7 from 2-chloro-4-(2-methyl-1H-imidazol-4-ylethynyl)-pyridine and 3-cyano-benzene boronic acid.

Sources & evidence

ORD record
ord-f6528944d4be4119b1810b906d177259
Source dataset
uspto-grants-2011_07
Patent number
US07973165B2

Reaction notes

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