HuagongsheHuagongshe Chemistry Print Report · For research reference only
(Pyrimidin-5-yl)boronic acid → HCID 49803714, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | (Pyrimidin-5-yl)boronic acid | HCID 2795193 | — |
| Reactant | HCID 49803415 | HCID 49803415 | — |
| Reactant | HCID 49803713 | HCID 49803713 | — |
| Product | HCID 49803714 | HCID 49803714 | 68% |
Reaction Steps
The procedure of Example 2 was repeated except for using N-(2-aminophenyl)-4-((4-bromo-1-oxoisoindolin-2-yl)methyl)benzamide in Example 9 instead of N-(2-aminophenyl)-4-((4-bromo-5,6-dimethoxy-1-oxoisoindolin-2-yl)methyl)benzamide, and pyrimidin-5-yl-5-boronic acid instead of phenyl boronic acid to obtain the title compound (68%).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08716326B2 |
| Source dataset | uspto-grants-2014_05 |
| ORD ID | ord-e41a2a8e274a4a18bd7bb9bb85238d0f |
| Source note | uspto-grants-2014_05 |